| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Free fatty acid receptor 4 |
|---|
| Ligand | BDBM382139 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | BRET assay |
|---|
| EC50 | 2750±n/a nM |
|---|
| Citation |  Kumar, S; Sharma, R; Deore, VB; Yewalkar, NN Substituted phenyl alkanoic acid compounds as GPR120 agonists and uses thereof US Patent US10273230 Publication Date 4/30/2019 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Free fatty acid receptor 4 |
|---|
| Name: | Free fatty acid receptor 4 |
|---|
| Synonyms: | FFAR4 | FFAR4_HUMAN | G-protein coupled receptor 120 | G-protein coupled receptor 129 | G-protein coupled receptor GT01 | G-protein coupled receptor PGR4 | GPR120 | GPR129 | O3FAR1 | Omega-3 fatty acid receptor 1 | PGR4 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 42256.91 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1508994 |
|---|
| Residue: | 377 |
|---|
| Sequence: | MSPECARAAGDAPLRSLEQANRTRFPFFSDVKGDHRLVLAAVETTVLVLIFAVSLLGNVC
ALVLVARRRRRGATACLVLNLFCADLLFISAIPLVLAVRWTEAWLLGPVACHLLFYVMTL
SGSVTILTLAAVSLERMVCIVHLQRGVRGPGRRARAVLLALIWGYSAVAALPLCVFFRVV
PQRLPGADQEISICTLIWPTIPGEISWDVSFVTLNFLVPGLVIVISYSKILQTSEHLLDA
RAVVTHSEITKASRKRLTVSLAYSESHQIRVSQQDFRLFRTLFLLMVSFFIMWSPIIITI
LLILIQNFKQDLVIWPSLFFWVVAFTFANSALNPILYNMTLCRNEWKKIFCCFWFPEKGA
ILTDTSVKRNDLSIISG
|
|
|
|---|
| BDBM382139 |
|---|
| n/a |
|---|
| Name | BDBM382139 |
|---|
| Synonyms: | 4-(4-((2-(p-tolyloxy)cyclohex-1-en-1-yl)methoxy)phenyl)butanoic Acid | US10273230, Compound of Example 50 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C24H28O4 |
|---|
| Mol. Mass. | 380.4767 |
|---|
| SMILES | Cc1ccc(OC2=C(COc3ccc(CCCC(O)=O)cc3)CCCC2)cc1 |c:6| |
|---|
| Structure | 
|
|---|
Search and Browse
