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TargetSerine/threonine-protein kinase pim-1
LigandBDBM26623
Substrate/CompetitorS6 kinase/Rsk-2 peptide 2
Meas. Tech.Pim Kinase Assay
pH7±n/a
Temperature298.15±n/a K
IC50 60±20 nM
Citation Xia, ZKnaak, CMa, JBeharry, ZMMcInnes, CWang, WKraft, ASSmith, CD Synthesis and evaluation of novel inhibitors of Pim-1 and Pim-2 protein kinases. J Med Chem52:74-86 (2009) [PubMed]  Article
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Serine/threonine-protein kinase pim-1
Name:Serine/threonine-protein kinase pim-1
Synonyms:PIM-1 Kinase | PIM1 | PIM1_HUMAN | Proto-oncogene serine/threonine-protein kinase Pim-1 | Serine/threonine-protein kinase (PIM1) | Serine/threonine-protein kinase PIM | Serine/threonine-protein kinase PIM1 | Serine/threonine-protein kinase pim-1 (PIM1)
Type:Protein
Mol. Mass.:35681.82
Organism:Homo sapiens (Human)
Description:P11309
Residue:313
Sequence:
MLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSD
NLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLIL
ERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRG
ELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDI
PFEHDEEIIRGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETA
EIHLHSLSPGPSK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM26623
S6 kinase/Rsk-2 peptide 2
Name:S6 kinase/Rsk-2 peptide 2
Synonyms:n/a
Type:Peptide
Mol. Mass.:1149.41
Organism:n/a
Description:n/a
Residue:9
Sequence:
KKRNRTLTK