| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Serine/threonine-protein kinase pim-2 |
|---|
| Ligand | BDBM26623 |
|---|
| Substrate/Competitor | S6 kinase/Rsk-2 peptide 2 |
|---|
| Meas. Tech. | Pim Kinase Assay |
|---|
| IC50 | 4400±n/a nM |
|---|
| Citation |  Xia, Z; Knaak, C; Ma, J; Beharry, ZM; McInnes, C; Wang, W; Kraft, AS; Smith, CD Synthesis and evaluation of novel inhibitors of Pim-1 and Pim-2 protein kinases. J Med Chem52:74-86 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Serine/threonine-protein kinase pim-2 |
|---|
| Name: | Serine/threonine-protein kinase pim-2 |
|---|
| Synonyms: | PIM2 | PIM2_HUMAN | Pim-2h | Serine/threonine-protein kinase (PIM2) | Serine/threonine-protein kinase PIM | Serine/threonine-protein kinase pim-2 (PIM2) |
|---|
| Type: | Serine/threonine-protein kinase |
|---|
| Mol. Mass.: | 34185.93 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q9P1W9 |
|---|
| Residue: | 311 |
|---|
| Sequence: | MLTKPLQGPPAPPGTPTPPPGGKDREAFEAEYRLGPLLGKGGFGTVFAGHRLTDRLQVAI
KVIPRNRVLGWSPLSDSVTCPLEVALLWKVGAGGGHPGVIRLLDWFETQEGFMLVLERPL
PAQDLFDYITEKGPLGEGPSRCFFGQVVAAIQHCHSRGVVHRDIKDENILIDLRRGCAKL
IDFGSGALLHDEPYTDFDGTRVYSPPEWISRHQYHALPATVWSLGILLYDMVCGDIPFER
DQEILEAELHFPAHVSPDCCALIRRCLAPKPSSRPSLEEILLDPWMQTPAEDVPLNPSKG
GPAPLAWSLLP
|
|
|
|---|
| BDBM26623 |
|---|
| S6 kinase/Rsk-2 peptide 2 |
|---|
| Name: | S6 kinase/Rsk-2 peptide 2 |
|---|
| Synonyms: | n/a |
|---|
| Type: | Peptide |
|---|
| Mol. Mass.: | 1149.41 |
|---|
| Organism: | n/a |
|---|
| Description: | n/a |
|---|
| Residue: | 9 |
|---|
| Sequence: | |
|---|
Search and Browse
