| Reaction Details |
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 | Report a problem with these data |
| Target | fMet-Leu-Phe receptor |
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| Ligand | BDBM37744 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands |
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| IC50 | 18400±n/a nM |
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| Citation |  PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| fMet-Leu-Phe receptor |
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| Name: | fMet-Leu-Phe receptor |
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| Synonyms: | FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38456.14 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_4503779 |
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| Residue: | 350 |
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| Sequence: | METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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| BDBM37744 |
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| n/a |
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| Name | BDBM37744 |
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| Synonyms: | 3-[2-(N-ethyl-2,5-dimethoxy-anilino)-2-keto-ethyl]-1H-indole-2-carboxylic acid | 3-[2-(N-ethyl-2,5-dimethoxyanilino)-2-oxoethyl]-1H-indole-2-carboxylic acid | 3-[2-[(2,5-dimethoxyphenyl)-ethyl-amino]-2-oxidanylidene-ethyl]-1H-indole-2-carboxylic acid | 3-{2-[(2,5-dimethoxyphenyl)(ethyl)amino]-2-oxoethyl}-1H-indole-2-carboxylic acid | MLS000044758 | SMR000022868 | cid_3244340 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H22N2O5 |
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| Mol. Mass. | 382.4098 |
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| SMILES | CCN(C(=O)Cc1c([nH]c2ccccc12)C(O)=O)c1cc(OC)ccc1OC |
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| Structure | 
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