| Reaction Details |
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 | Report a problem with these data |
| Target | fMet-Leu-Phe receptor |
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| Ligand | BDBM37771 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands |
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| IC50 | 15300±n/a nM |
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| Citation |  PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| fMet-Leu-Phe receptor |
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| Name: | fMet-Leu-Phe receptor |
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| Synonyms: | FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38456.14 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_4503779 |
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| Residue: | 350 |
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| Sequence: | METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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| BDBM37771 |
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| n/a |
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| Name | BDBM37771 |
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| Synonyms: | 2-(4-ethoxyphenyl)-3-(furan-2-carbonyl)-4-hydroxy-1-(pyridin-3-ylmethyl)-2H-pyrrol-5-one | 2-(4-ethoxyphenyl)-3-(furan-2-ylcarbonyl)-4-oxidanyl-1-(pyridin-3-ylmethyl)-2H-pyrrol-5-one | 2-(4-ethoxyphenyl)-3-[2-furanyl(oxo)methyl]-4-hydroxy-1-(3-pyridinylmethyl)-2H-pyrrol-5-one | 4-(2-furoyl)-3-hydroxy-5-p-phenetyl-1-(3-pyridylmethyl)-3-pyrrolin-2-one | 5-(4-ethoxyphenyl)-4-(2-furoyl)-3-hydroxy-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one | MLS000063148 | SMR000071444 | cid_2919194 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H20N2O5 |
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| Mol. Mass. | 404.4153 |
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| SMILES | CCOc1ccc(cc1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1Cc1cccnc1 |
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| Structure | 
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