Reaction Details |
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Target | fMet-Leu-Phe receptor |
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Ligand | BDBM37812 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands |
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IC50 | 27000±n/a nM |
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Citation | PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay(2007)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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fMet-Leu-Phe receptor |
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Name: | fMet-Leu-Phe receptor |
Synonyms: | FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 38456.14 |
Organism: | Homo sapiens (Human) |
Description: | gi_4503779 |
Residue: | 350 |
Sequence: | METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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BDBM37812 |
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n/a |
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Name | BDBM37812 |
Synonyms: | 1-(2-furanylmethyl)-4-hydroxy-3-[oxo(thiophen-2-yl)methyl]-2-(3,4,5-trimethoxyphenyl)-2H-pyrrol-5-one | 1-(2-furfuryl)-3-hydroxy-4-(2-thenoyl)-5-(3,4,5-trimethoxyphenyl)-3-pyrrolin-2-one | 1-(furan-2-ylmethyl)-4-hydroxy-3-(thiophene-2-carbonyl)-2-(3,4,5-trimethoxyphenyl)-2H-pyrrol-5-one | 1-(furan-2-ylmethyl)-4-oxidanyl-3-thiophen-2-ylcarbonyl-2-(3,4,5-trimethoxyphenyl)-2H-pyrrol-5-one | MLS000113983 | SMR000109873 | cid_2934026 |
Type | Small organic molecule |
Emp. Form. | C23H21NO7S |
Mol. Mass. | 455.48 |
SMILES | COc1cc(cc(OC)c1OC)C1C(C(=O)c2cccs2)C(=O)C(=O)N1Cc1ccco1 |
Structure |
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