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Reaction Details
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TargetN-formyl peptide receptor 2
LigandBDBM40450
Substrate/Competitorn/a
Meas. Tech.Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1)
IC50>66700±n/a nM
Citation PubChem, PC Formylpeptide Receptor (FPR) Ligand Structure Activity Relationship (SAR) Analysis : Dose Response Assay Counterscreen Against Formyl Peptide Receptor-Like-1 (FPRL1)  PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
N-formyl peptide receptor 2
Name:N-formyl peptide receptor 2
Synonyms:ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:38968.35
Organism:Homo sapiens (Human)
Description:P25090
Residue:351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVT
TICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIA
LDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNF
ASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPL
RVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPM
LYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
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  Blast E-value cutoff:
BDBM40450
n/a
NameBDBM40450
Synonyms:N-(2,6-dimethylphenyl)-2-[(1-oxo-2-thiophen-2-ylethyl)amino]-2-phenylacetamide | N-(2,6-dimethylphenyl)-2-phenyl-2-(2-thiophen-2-ylethanoylamino)ethanamide | N-(2,6-dimethylphenyl)-2-phenyl-2-[(2-thiophen-2-ylacetyl)amino]acetamide | N-(2,6-dimethylphenyl)-2-phenyl-2-[[2-(2-thienyl)acetyl]amino]acetamide | UNM000003608101 | cid_4656066
TypeSmall organic molecule
Emp. Form.C22H22N2O2S
Mol. Mass.378.487
SMILESCc1cccc(C)c1NC(=O)C(NC(=O)Cc1cccs1)c1ccccc1
Structure
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