Ki Summary

Reaction Details

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Target

Nuclear receptor subfamily 4 group A member 1

Ligand

BDBM40630

Substrate/Competitor

n/a

Meas. Tech.

High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters

IC50

12555±2050 nM

Citation

PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Nuclear receptor subfamily 4 group A member 1

Name:

Nuclear receptor subfamily 4 group A member 1

Synonyms:

GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1

Type:

Enzyme Catalytic Domain

Mol. Mass.:

64467.13

Organism:

Homo sapiens (Human)

Description:

gi_27894344

Residue:

598

Sequence:

MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF

BDBM40630

n/a

Name

BDBM40630

Synonyms:

MLS000087341 | N-(2-methylsulfanylphenyl)-5,6-dihydro-4H-cyclopenta[d][1,2]oxazole-3-carboxamide | N-[2-(methylthio)phenyl]-5,6-dihydro-4H-cyclopent[d]isoxazole-3-carboxamide | N-[2-(methylthio)phenyl]-5,6-dihydro-4H-cyclopenta[d]isoxazole-3-carboxamide | SMR000023564 | cid_3238925

Type

Small organic molecule

Emp. Form.

C14H14N2O2S

Mol. Mass.

274.338

SMILES

CSc1ccccc1NC(=O)c1noc2CCCc12

Structure