Ki Summary

Reaction Details

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Target

Nuclear receptor subfamily 4 group A member 1

Ligand

BDBM40639

Substrate/Competitor

n/a

Meas. Tech.

High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters

IC50

558.14±88 nM

Citation

PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Nuclear receptor subfamily 4 group A member 1

Name:

Nuclear receptor subfamily 4 group A member 1

Synonyms:

GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1

Type:

Enzyme Catalytic Domain

Mol. Mass.:

64467.13

Organism:

Homo sapiens (Human)

Description:

gi_27894344

Residue:

598

Sequence:

MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF

BDBM40639

n/a

Name

BDBM40639

Synonyms:

3-bromanyl-4-ethoxy-N-[4-(4-methylpiperazin-1-yl)phenyl]benzamide | 3-bromo-4-ethoxy-N-[4-(4-methyl-1-piperazinyl)phenyl]benzamide | 3-bromo-4-ethoxy-N-[4-(4-methylpiperazin-1-yl)phenyl]benzamide | 3-bromo-4-ethoxy-N-[4-(4-methylpiperazino)phenyl]benzamide | MLS000049130 | SMR000074453 | cid_1017508

Type

Small organic molecule

Emp. Form.

C20H24BrN3O2

Mol. Mass.

418.327

SMILES

CCOc1ccc(cc1Br)C(=O)Nc1ccc(cc1)N1CCN(C)CC1

Structure