Reaction Details |
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Target | Nuclear receptor subfamily 4 group A member 1 |
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Ligand | BDBM40727 |
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Substrate/Competitor | n/a |
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Meas. Tech. | High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters |
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IC50 | 2965.6±99.3 nM |
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Citation | PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Nuclear receptor subfamily 4 group A member 1 |
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Name: | Nuclear receptor subfamily 4 group A member 1 |
Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 64467.13 |
Organism: | Homo sapiens (Human) |
Description: | gi_27894344 |
Residue: | 598 |
Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
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BDBM40727 |
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n/a |
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Name | BDBM40727 |
Synonyms: | MLS000537135 | N'-(4-fluorobenzylidene)-2-(2-furyl)-4-quinolinecarbohydrazide | N-[(4-fluorobenzylidene)amino]-2-(2-furyl)cinchoninamide | N-[(4-fluorophenyl)methylideneamino]-2-(2-furanyl)-4-quinolinecarboxamide | N-[(4-fluorophenyl)methylideneamino]-2-(furan-2-yl)quinoline-4-carboxamide | SMR000159894 | cid_1226487 |
Type | Small organic molecule |
Emp. Form. | C21H14FN3O2 |
Mol. Mass. | 359.3532 |
SMILES | Fc1ccc(C=NNC(=O)c2cc(nc3ccccc23)-c2ccco2)cc1 |w:6.6| |
Structure |
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