Ki Summary

Reaction Details

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Target

Sphingosine 1-phosphate receptor 2

Ligand

BDBM41584

Substrate/Competitor

n/a

Meas. Tech.

Dose Response Cell Based Assay for Antagonists of the S1P2 Receptor

IC50

2943±n/a nM

Citation

PubChem, PC Dose Response Cell Based Assay for Antagonists of the S1P2 Receptor PubChem Bioassay(2007)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Sphingosine 1-phosphate receptor 2

Name:

Sphingosine 1-phosphate receptor 2

Synonyms:

Type:

G Protein-Coupled Receptor (GPCR)

Mol. Mass.:

38883.16

Organism:

Homo sapiens (Human)

Description:

Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay.

Residue:

353

Sequence:

MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVAR
NSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASV
FSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACS
TVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLG
VFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVL
RPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV

BDBM41584

n/a

Name

BDBM41584

Synonyms:

(4-decyl-1,2,3,5,6,7-hexahydrodicyclopenta[1,2-c:1',2'-g]pyridin-8-ylidene)amine;hydrobromide | 4-Decyl-2,3,4,5,6,7-hexahydro-1H-4-aza-s-indacen-8-ylideneamine | 4-decyl-1,2,3,5,6,7-hexahydrodicyclopenta[1,2-c:1',2'-g]pyridin-8-imine;hydrobromide | MLS000525289 | SMR000122163 | cid_9549474

Type

Small organic molecule

Emp. Form.

C21H34N2

Mol. Mass.

314.5081

SMILES

CCCCCCCCCCn1c2CCCc2c(=N)c2CCCc12

Structure