| Reaction Details |
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 | Report a problem with these data |
| Target | Sphingosine 1-phosphate receptor 2 |
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| Ligand | BDBM39773 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response Cell Based Assay for Antagonists of the S1P2 Receptor |
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| IC50 | 2939±n/a nM |
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| Citation |  PubChem, PC Dose Response Cell Based Assay for Antagonists of the S1P2 Receptor PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Sphingosine 1-phosphate receptor 2 |
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| Name: | Sphingosine 1-phosphate receptor 2 |
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| Synonyms: | EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 38883.16 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay. |
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| Residue: | 353 |
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| Sequence: | MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVAR
NSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASV
FSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACS
TVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLG
VFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVL
RPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
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| BDBM39773 |
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| n/a |
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| Name | BDBM39773 |
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| Synonyms: | (2Z)-3-ethyl-2-[(1-ethyl-8-methyl-2-quinolin-1-iumyl)methylidene]-1,3-benzothiazole;iodide | (2Z)-3-ethyl-2-[(1-ethyl-8-methyl-quinolin-1-ium-2-yl)methylene]-1,3-benzothiazole;iodide | (2Z)-3-ethyl-2-[(1-ethyl-8-methyl-quinolin-1-ium-2-yl)methylidene]-1,3-benzothiazole;iodide | (2Z)-3-ethyl-2-[(1-ethyl-8-methylquinolin-1-ium-2-yl)methylidene]-1,3-benzothiazole;iodide | 1-Ethyl-2-(3-ethyl-3H-benzothiazol-2-ylidenemethyl)-8-methyl-quinolinium | MLS000556089 | SMR000177972 | cid_11958727 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H23N2S |
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| Mol. Mass. | 347.496 |
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| SMILES | CCN1\C(Sc2ccccc12)=C\c1ccc2cccc(C)c2[n+]1CC |
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| Structure | 
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