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TargetSphingosine 1-phosphate receptor 2
LigandBDBM41658
Substrate/Competitorn/a
Meas. Tech.Dose Response Cell Based Assay for Agonists of the S1P2 Receptor
EC50>50000±n/a nM
Citation PubChem, PC Dose Response Cell Based Assay for Agonists of the S1P2 Receptor PubChem Bioassay(2007)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Sphingosine 1-phosphate receptor 2
Name:Sphingosine 1-phosphate receptor 2
Synonyms:EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:38883.16
Organism:Homo sapiens (Human)
Description:Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay.
Residue:353
Sequence:
MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVAR
NSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASV
FSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACS
TVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLG
VFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVL
RPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM41658
n/a
NameBDBM41658
Synonyms:1-(4-chlorophenyl)-N-(2-oxolanylmethyl)methanesulfonamide | 1-(4-chlorophenyl)-N-(oxolan-2-ylmethyl)methanesulfonamide | 1-(4-chlorophenyl)-N-(tetrahydro-2-furanylmethyl)methanesulfonamide | 1-(4-chlorophenyl)-N-(tetrahydrofurfuryl)methanesulfonamide | MLS000099995 | SMR000081216 | cid_2973451
TypeSmall organic molecule
Emp. Form.C12H16ClNO3S
Mol. Mass.289.778
SMILESClc1ccc(CS(=O)(=O)NCC2CCCO2)cc1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: