Ki Summary

Reaction Details

Report a problem with these data

Target

Nuclear receptor subfamily 4 group A member 1

Ligand

BDBM42084

Substrate/Competitor

n/a

Meas. Tech.

Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors

EC50

5700±5960 nM

Citation

PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Nuclear receptor subfamily 4 group A member 1

Name:

Nuclear receptor subfamily 4 group A member 1

Synonyms:

GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1

Type:

Enzyme Catalytic Domain

Mol. Mass.:

64467.13

Organism:

Homo sapiens (Human)

Description:

gi_27894344

Residue:

598

Sequence:

MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF

BDBM42084

n/a

Name

BDBM42084

Synonyms:

2-[(Z)-1-nitro-2-[(phenylmethyl)amino]ethenyl]cyclohexa-2,5-diene-1,4-dione | 2-[(Z)-2-(benzylamino)-1-nitro-vinyl]-p-benzoquinone | 2-[(Z)-2-(benzylamino)-1-nitroethenyl]cyclohexa-2,5-diene-1,4-dione | BIM-0048185.P001 | cid_792475

Type

Small organic molecule

Emp. Form.

C15H12N2O4

Mol. Mass.

284.2668

SMILES

[O-][N+](=O)C(C=NCc1ccccc1)C1=CC(=O)C=CC1=O |w:5.5,c:18,t:14|

Structure