Ki Summary

Reaction Details

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Target

Nuclear receptor subfamily 4 group A member 1

Ligand

BDBM42090

Substrate/Competitor

n/a

Meas. Tech.

Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors

EC50

4390±7210 nM

Citation

PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Nuclear receptor subfamily 4 group A member 1

Name:

Nuclear receptor subfamily 4 group A member 1

Synonyms:

GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1

Type:

Enzyme Catalytic Domain

Mol. Mass.:

64467.13

Organism:

Homo sapiens (Human)

Description:

gi_27894344

Residue:

598

Sequence:

MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF

BDBM42090

n/a

Name

BDBM42090

Synonyms:

1-(2-pyridinyl)-N-[4-(2-pyridinylmethylideneamino)phenyl]methanimine | 1-pyridin-2-yl-N-[4-(pyridin-2-ylmethylideneamino)phenyl]methanimine | 2-pyridylmethylene-[4-(2-pyridylmethyleneamino)phenyl]amine | BIM-0022469.P001 | cid_870650

Type

Small organic molecule

Emp. Form.

C18H14N4

Mol. Mass.

286.3306

SMILES

C(=N/c1ccc(cc1)\N=C\c1ccccn1)\c1ccccn1

Structure