BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetNuclear receptor subfamily 4 group A member 1
LigandBDBM42094
Substrate/Competitorn/a
Meas. Tech.Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors
EC50 14400±20590 nM
Citation PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Nuclear receptor subfamily 4 group A member 1
Name:Nuclear receptor subfamily 4 group A member 1
Synonyms:GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1
Type:Enzyme Catalytic Domain
Mol. Mass.:64467.13
Organism:Homo sapiens (Human)
Description:gi_27894344
Residue:598
Sequence:
MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM42094
n/a
NameBDBM42094
Synonyms:2-[[1-(4-chlorobenzyl)indol-3-yl]methylene]indane-1,3-quinone | 2-[[1-[(4-chlorophenyl)methyl]-3-indolyl]methylidene]indene-1,3-dione | 2-[[1-[(4-chlorophenyl)methyl]indol-3-yl]methylidene]indene-1,3-dione | BIM-0025627.P001 | cid_1118107
TypeSmall organic molecule
Emp. Form.C25H16ClNO2
Mol. Mass.397.853
SMILESClc1ccc(-[#6]-n2cc(\[#6]=[#6]-3/[#6](=O)-c4ccccc4-[#6]-3=O)c3ccccc23)cc1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: