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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Nuclear receptor subfamily 4 group A member 1 | ||
| Ligand | BDBM42097 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors | ||
| EC50 | 23760±19510 nM | ||
| Citation |  PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| Nuclear receptor subfamily 4 group A member 1 | |||
| Name: | Nuclear receptor subfamily 4 group A member 1 | ||
| Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 64467.13 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | gi_27894344 | ||
| Residue: | 598 | ||
| Sequence: |
| ||
| BDBM42097 | |||
| n/a | |||
| Name | BDBM42097 | ||
| Synonyms: | 1',3'-bis(oxidanyl)spiro[2,5-dihydro-[1,2,4]triazolo[4,3-b][1,2,4,5]tetrazine-6,2'-indene]-3-thione | 1',3'-dihydroxy-3-spiro[2,5-dihydro-[1,2,4]triazolo[4,3-b][1,2,4,5]tetrazine-6,2'-indene]thione | 1',3'-dihydroxyspiro[2,5-dihydro-[1,2,4]triazolo[4,3-b][1,2,4,5]tetrazine-6,2'-indene]-3-thione | BIM-0026580.P001 | cid_5341377 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C11H8N6O2S | ||
| Mol. Mass. | 288.285 | ||
| SMILES | OC1c2ccccc2C(=O)C11Nn2c(n[nH]c2=S)N=N1 |c:21| | ||
| Structure | 
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