| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 4 group A member 1 |
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| Ligand | BDBM42108 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors |
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| EC50 | 33360±66780 nM |
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| Citation |  PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Nuclear receptor subfamily 4 group A member 1 |
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| Name: | Nuclear receptor subfamily 4 group A member 1 |
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| Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 64467.13 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_27894344 |
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| Residue: | 598 |
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| Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
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| BDBM42108 |
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| n/a |
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| Name | BDBM42108 |
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| Synonyms: | (4Z)-1-(3-chloranyl-4-fluoranyl-phenyl)-4-(furan-2-ylmethylidene)pyrazolidine-3,5-dione | (4Z)-1-(3-chloro-4-fluoro-phenyl)-4-(2-furfurylidene)pyrazolidine-3,5-quinone | (4Z)-1-(3-chloro-4-fluorophenyl)-4-(2-furanylmethylidene)pyrazolidine-3,5-dione | (4Z)-1-(3-chloro-4-fluorophenyl)-4-(furan-2-ylmethylidene)pyrazolidine-3,5-dione | BIM-0049357.P001 | cid_5343905 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H8ClFN2O3 |
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| Mol. Mass. | 306.676 |
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| SMILES | Fc1ccc(cc1Cl)N1NC(=O)\C(=C\c2ccco2)C1=O |
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| Structure | 
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