| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Nuclear receptor subfamily 4 group A member 1 |
|---|
| Ligand | BDBM42111 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors |
|---|
| EC50 | 4950±5280 nM |
|---|
| Citation |  PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Nuclear receptor subfamily 4 group A member 1 |
|---|
| Name: | Nuclear receptor subfamily 4 group A member 1 |
|---|
| Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 64467.13 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_27894344 |
|---|
| Residue: | 598 |
|---|
| Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
|
|
|
|---|
| BDBM42111 |
|---|
| n/a |
|---|
| Name | BDBM42111 |
|---|
| Synonyms: | 6-(pyrrolidine-1-carbonyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid | 6-[oxo(1-pyrrolidinyl)methyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid | 6-pyrrolidin-1-ylcarbonyl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid | BIM-0049524.P001 | cid_3955075 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H20N2O3 |
|---|
| Mol. Mass. | 312.363 |
|---|
| SMILES | OC(=O)C1Nc2c(cccc2C(=O)N2CCCC2)C2C=CCC12 |c:21| |
|---|
| Structure | 
|
|---|
Search and Browse
