Ki Summary

Reaction Details

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Target

Nuclear receptor subfamily 4 group A member 1

Ligand

BDBM42119

Substrate/Competitor

n/a

Meas. Tech.

Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors

EC50

8750±2810 nM

Citation

PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Nuclear receptor subfamily 4 group A member 1

Name:

Nuclear receptor subfamily 4 group A member 1

Synonyms:

GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1

Type:

Enzyme Catalytic Domain

Mol. Mass.:

64467.13

Organism:

Homo sapiens (Human)

Description:

gi_27894344

Residue:

598

Sequence:

MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF

BDBM42119

n/a

Name

BDBM42119

Synonyms:

2-[4-(2,5-dimethyl-1-pyrrolyl)phenoxy]acetic acid | 2-[4-(2,5-dimethylpyrrol-1-yl)phenoxy]acetic acid | 2-[4-(2,5-dimethylpyrrol-1-yl)phenoxy]ethanoic acid | BIM-0001419.P001 | cid_776871

Type

Small organic molecule

Emp. Form.

C14H15NO3

Mol. Mass.

245.2738

SMILES

Cc1ccc(C)n1-c1ccc(OCC(O)=O)cc1

Structure