| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 4 group A member 1 |
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| Ligand | BDBM15186 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors |
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| EC50 | 1650±450 nM |
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| Citation |  PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Nuclear receptor subfamily 4 group A member 1 |
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| Name: | Nuclear receptor subfamily 4 group A member 1 |
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| Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 64467.13 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_27894344 |
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| Residue: | 598 |
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| Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
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| BDBM15186 |
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| n/a |
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| Name | BDBM15186 |
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| Synonyms: | 4-(5-{[(5E)-2-amino-3,7-dicyano-4,6-dimethyl-5H-cyclopenta[b]pyridin-5-ylidene]methyl}furan-2-yl)-2-chlorobenzoic acid | cid_1776570 | compound 1 | compound 6065233 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H15ClN4O3 |
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| Mol. Mass. | 442.854 |
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| SMILES | Cc1c(C#N)c(N)[nH]c2c(C#N)c(=C)c(=Cc3ccc(o3)-c3ccc(C(O)=O)c(Cl)c3)c12 |w:15.15| |
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| Structure | 
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