Reaction Details |
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Target | Nuclear receptor subfamily 4 group A member 1 |
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Ligand | BDBM42123 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors |
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EC50 | 3740±5300 nM |
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Citation | PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Nuclear receptor subfamily 4 group A member 1 |
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Name: | Nuclear receptor subfamily 4 group A member 1 |
Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 64467.13 |
Organism: | Homo sapiens (Human) |
Description: | gi_27894344 |
Residue: | 598 |
Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
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BDBM42123 |
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n/a |
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Name | BDBM42123 |
Synonyms: | BIM-0013886.P001 | cid_878844 |
Type | Small organic molecule |
Emp. Form. | C13H9N5 |
Mol. Mass. | 235.2441 |
SMILES | Nc1[nH]nc2ncc3cc4ccccc4nc3c12 |
Structure |
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