| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 4 group A member 1 |
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| Ligand | BDBM42124 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors |
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| EC50 | 12900±10180 nM |
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| Citation |  PubChem, PC Fluorescence Polarization Dose Response Assay for TR3-Based Bcl-B Inhibitors PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Nuclear receptor subfamily 4 group A member 1 |
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| Name: | Nuclear receptor subfamily 4 group A member 1 |
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| Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 64467.13 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_27894344 |
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| Residue: | 598 |
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| Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
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| BDBM42124 |
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| n/a |
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| Name | BDBM42124 |
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| Synonyms: | 2-(1,3-benzothiazol-2-ylsulfanyl)-N-[(Z)-[1-[(4-methylpiperazin-1-yl)methyl]-2-oxidanylidene-indol-3-ylidene]amino]ethanamide | 2-(1,3-benzothiazol-2-ylsulfanyl)-N-[(Z)-[1-[(4-methylpiperazin-1-yl)methyl]-2-oxoindol-3-ylidene]amino]acetamide | 2-(1,3-benzothiazol-2-ylthio)-N-[(Z)-[1-[(4-methyl-1-piperazinyl)methyl]-2-oxo-3-indolylidene]amino]acetamide | 2-(1,3-benzothiazol-2-ylthio)-N-[(Z)-[2-keto-1-[(4-methylpiperazino)methyl]indolin-3-ylidene]amino]acetamide | BIM-0043480.P001 | cid_5347365 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H24N6O2S2 |
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| Mol. Mass. | 480.606 |
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| SMILES | CN1CCN(CN2C(=O)\C(=N/NC(=O)CSc3nc4ccccc4s3)c3ccccc23)CC1 |
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| Structure | 
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