| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 1 |
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| Ligand | BDBM42498 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism |
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| IC50 | 6433±n/a nM |
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| Citation |  PubChem, PC Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Neuropeptide Y receptor type 1 |
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| Name: | Neuropeptide Y receptor type 1 |
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| Synonyms: | NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44399.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | NPY-Y1 NPY1R HUMAN::P25929 |
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| Residue: | 384 |
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| Sequence: | MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLA
LIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQ
CVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMT
DEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKR
RNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNL
LFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVS
KTSLKQASPVAFKKINNNDDNEKI
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| BDBM42498 |
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| n/a |
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| Name | BDBM42498 |
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| Synonyms: | MLS000520555 | N-[2-[4-(2,3-dimethylphenyl)-1-piperazinyl]ethyl]-2-[2-[(2-methylphenyl)-oxomethyl]-1-pyrrolyl]acetamide | N-[2-[4-(2,3-dimethylphenyl)piperazin-1-yl]ethyl]-2-[2-(2-methylbenzoyl)pyrrol-1-yl]acetamide | N-[2-[4-(2,3-dimethylphenyl)piperazin-1-yl]ethyl]-2-[2-(2-methylphenyl)carbonylpyrrol-1-yl]ethanamide | N-[2-[4-(2,3-dimethylphenyl)piperazino]ethyl]-2-(2-o-toluoylpyrrol-1-yl)acetamide | SMR000130966 | cid_9550576 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H34N4O2 |
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| Mol. Mass. | 458.5952 |
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| SMILES | Cc1cccc(N2CCN(CCNC(=O)Cn3cccc3C(=O)c3ccccc3C)CC2)c1C |
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| Structure | 
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