Ki Summary

Reaction Details

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Target

Neuropeptide Y receptor type 1

Ligand

BDBM42568

Substrate/Competitor

n/a

Meas. Tech.

Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism

IC50

5853±n/a nM

Citation

PubChem, PC Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism PubChem Bioassay(2008)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Neuropeptide Y receptor type 1

Name:

Neuropeptide Y receptor type 1

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

44399.07

Organism:

Homo sapiens (Human)

Description:

NPY-Y1 NPY1R HUMAN::P25929

Residue:

384

Sequence:

MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLA
LIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQ
CVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMT
DEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKR
RNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNL
LFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVS
KTSLKQASPVAFKKINNNDDNEKI

BDBM42568

n/a

Name

BDBM42568

Synonyms:

(Z)-2-methyl-2-butenoic acid [(8S,9R)-8-[2-[(Z)-2-methyl-1-oxobut-2-enoxy]propan-2-yl]-2-oxo-8,9-dihydrofuro[2,3-h][1]benzopyran-9-yl] ester | (Z)-2-methylbut-2-enoic acid [(8S,9R)-2-keto-8-[1-methyl-1-[(Z)-2-methylbut-2-enoyl]oxy-ethyl]-8,9-dihydrofuro[2,3-h]chromen-9-yl] ester | MLS000574899 | SMR000156245 | [(8S,9R)-8-[2-[(Z)-2-methylbut-2-enoyl]oxypropan-2-yl]-2-oxidanylidene-8,9-dihydrofuro[2,3-h]chromen-9-yl] (Z)-2-methylbut-2-enoate | [(8S,9R)-8-[2-[(Z)-2-methylbut-2-enoyl]oxypropan-2-yl]-2-oxo-8,9-dihydrofuro[2,3-h]chromen-9-yl] (Z)-2-methylbut-2-enoate | cid_5281371

Type

Small organic molecule

Emp. Form.

C24H26O7

Mol. Mass.

426.459

SMILES

C\C=C(\C)C(=O)O[C@H]1[C@H](Oc2ccc3ccc(=O)oc3c12)C(C)(C)OC(=O)C(\C)=C/C

Structure