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TargetCell division control protein 42 homolog
LigandBDBM43227
Substrate/Competitorn/a
Meas. Tech.Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant
EC50 11340±n/a nM
Citation PubChem, PC Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cell division control protein 42 homolog
Name:Cell division control protein 42 homolog
Synonyms:CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa)
Type:PROTEIN
Mol. Mass.:21258.36
Organism:Homo sapiens (Human)
Description:ChEMBL_652970
Residue:191
Sequence:
MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
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BDBM43227
n/a
NameBDBM43227
Synonyms:1-[2-(4-chlorophenyl)ethylamino]-3-(2-naphthalenyloxy)-2-propanol | 1-[2-(4-chlorophenyl)ethylamino]-3-(2-naphthoxy)propan-2-ol | 1-[2-(4-chlorophenyl)ethylamino]-3-naphthalen-2-yloxy-propan-2-ol | 1-[2-(4-chlorophenyl)ethylamino]-3-naphthalen-2-yloxypropan-2-ol | MLS000772350 | SMR000344505 | cid_4388447
TypeSmall organic molecule
Emp. Form.C21H22ClNO2
Mol. Mass.355.858
SMILESOC(CNCCc1ccc(Cl)cc1)COc1ccc2ccccc2c1
Structure
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