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TargetCell division control protein 42 homolog
LigandBDBM43236
Substrate/Competitorn/a
Meas. Tech.Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant
EC50 18690±n/a nM
Citation PubChem, PC Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Cdc42 activated mutant PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Cell division control protein 42 homolog
Name:Cell division control protein 42 homolog
Synonyms:CDC42 | CDC42_HUMAN | Cell division control protein 42 homolog | G25K GTP-binding protein | cell division cycle 42 (GTP binding protein, 25kDa)
Type:PROTEIN
Mol. Mass.:21258.36
Organism:Homo sapiens (Human)
Description:ChEMBL_652970
Residue:191
Sequence:
MQTIKCVVVGDGAVGKTCLLISYTTNKFPSEYVPTVFDNYAVTVMIGGEPYTLGLFDTAG
QEDYDRLRPLSYPQTDVFLVCFSVVSPSSFENVKEKWVPEITHHCPKTPFLLVGTQIDLR
DDPSTIEKLAKNKQKPITPETAEKLARDLKAVKYVECSALTQKGLKNVFDEAILAALEPP
EPKKSRRCVLL
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BDBM43236
n/a
NameBDBM43236
Synonyms:2-(4-chlorophenyl)sulfanylquinoline-4-carboxylic acid | 2-[(4-chlorophenyl)thio]-4-quinolinecarboxylic acid | 2-[(4-chlorophenyl)thio]cinchoninic acid | UNM000011083801 | cid_4550953
TypeSmall organic molecule
Emp. Form.C16H10ClNO2S
Mol. Mass.315.774
SMILESOC(=O)c1cc(Sc2ccc(Cl)cc2)nc2ccccc12
Structure
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