| Reaction Details |
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 | Report a problem with these data |
| Target | Ras-related protein Rab-2A |
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| Ligand | BDBM43233 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rab2 wildtype |
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| EC50 | 4877±n/a nM |
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| Citation |  PubChem, PC Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rab2 wildtype PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Ras-related protein Rab-2A |
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| Name: | Ras-related protein Rab-2A |
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| Synonyms: | RAB2 | RAB2A | RAB2A_CANLF | Ras-related protein Rab-2A. |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 23545.28 |
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| Organism: | Canis lupus familiaris |
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| Description: | gi_46577642 |
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| Residue: | 212 |
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| Sequence: | MAYAYLFKYIIIGDTGVGKSCLLLQFTDKRFQPVHDLTIGVEFGARMITIDGKQIKLQIW
DTAGQESFRSITRSYYRGAAGALLVYDITRRDTFNHLTTWLEDARQHSNSNMVIMLIGNK
SDLESRREVKKEEGEAFAREHGLIFMETSAKTASNVEEAFINTAKEIYEKIQEGVFDINN
EANGIKIGPQHAATNATHAGNQGGQQAGGGCC
|
|
|
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| BDBM43233 |
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| n/a |
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| Name | BDBM43233 |
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| Synonyms: | 1-benzyl-5-chloro-3-methyl-pyrazole-4-carboxylic acid | 1-benzyl-5-chloro-3-methylpyrazole-4-carboxylic acid | 5-chloranyl-3-methyl-1-(phenylmethyl)pyrazole-4-carboxylic acid | 5-chloro-3-methyl-1-(phenylmethyl)-4-pyrazolecarboxylic acid | MLS000759940 | SMR000370104 | cid_2393574 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H11ClN2O2 |
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| Mol. Mass. | 250.681 |
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| SMILES | Cc1nn(Cc2ccccc2)c(Cl)c1C(O)=O |
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| Structure | 
|
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