Reaction Details |
![](/images/Email.png) | Report a problem with these data |
Target | Signal transducer and activator of transcription 3 [702-738,740-752] |
---|
Ligand | BDBM43615 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | Dose response cell-based assay to measure STAT3 activation |
---|
IC50 | 3325±n/a nM |
---|
Citation | PubChem, PC Dose response cell-based assay to measure STAT3 activation PubChem Bioassay(2008)[AID] |
---|
More Info.: | Get all data from this article, Solution Info, Assay Method |
---|
|
Signal transducer and activator of transcription 3 [702-738,740-752] |
---|
Name: | Signal transducer and activator of transcription 3 [702-738,740-752] |
Synonyms: | APRF | STAT3 | STAT3_HUMAN |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 5263.93 |
Organism: | Homo sapiens (Human) |
Description: | gi_13272532 |
Residue: | 50 |
Sequence: | AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
|
|
|
BDBM43615 |
---|
n/a |
---|
Name | BDBM43615 |
Synonyms: | 2-(2-keto-4-methyl-pyrimid[1,2-b]indazol-6-yl)-N-propyl-acetamide | 2-(4-methyl-2-oxidanylidene-pyrimido[1,2-b]indazol-6-yl)-N-propyl-ethanamide | 2-(4-methyl-2-oxo-6-pyrimido[1,2-b]indazolyl)-N-propylacetamide | 2-(4-methyl-2-oxopyrimido[1,2-b]indazol-6-yl)-N-propylacetamide | MLS000522787 | SMR000128053 | cid_3249106 |
Type | Small organic molecule |
Emp. Form. | C16H18N4O2 |
Mol. Mass. | 298.3397 |
SMILES | CCCNC(=O)Cn1c2ccccc2c2nc(=O)cc(C)n12 |
Structure |
|