| Reaction Details |
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 | Report a problem with these data |
| Target | Signal transducer and activator of transcription 3 [702-738,740-752] |
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| Ligand | BDBM43516 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response counterscreen for STAT1 inhibitors: cell-based high throughput assay to measure STAT3 inhibition |
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| IC50 | >55700±n/a nM |
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| Citation |  PubChem, PC Dose response counterscreen for STAT1 inhibitors: cell-based high throughput assay to measure STAT3 inhibition PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Signal transducer and activator of transcription 3 [702-738,740-752] |
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| Name: | Signal transducer and activator of transcription 3 [702-738,740-752] |
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| Synonyms: | APRF | STAT3 | STAT3_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 5263.93 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_13272532 |
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| Residue: | 50 |
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| Sequence: | AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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| BDBM43516 |
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| n/a |
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| Name | BDBM43516 |
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| Synonyms: | 3-(anilinosulfonyl)-4-methyl-N-{3-[methyl(methylsulfonyl)amino]phenyl}benzamide | 4-methyl-N-[3-[methyl(methylsulfonyl)amino]phenyl]-3-(phenylsulfamoyl)benzamide | MLS000582661 | N-[3-[mesyl(methyl)amino]phenyl]-4-methyl-3-(phenylsulfamoyl)benzamide | SMR000201362 | cid_2231989 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H23N3O5S2 |
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| Mol. Mass. | 473.565 |
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| SMILES | CN(c1cccc(NC(=O)c2ccc(C)c(c2)S(=O)(=O)Nc2ccccc2)c1)S(C)(=O)=O |
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| Structure | 
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