| Reaction Details |
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 | Report a problem with these data |
| Target | Dual specificity protein phosphatase 3 |
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| Ligand | BDBM46286 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR VHR1 Fluorescent Assay for In Vitro dose response studies |
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| IC50 | 14000±n/a nM |
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| Citation |  PubChem, PC SAR VHR1 Fluorescent Assay for In Vitro dose response studies PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Dual specificity protein phosphatase 3 |
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| Name: | Dual specificity protein phosphatase 3 |
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| Synonyms: | DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR |
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| Type: | Hydrolase |
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| Mol. Mass.: | 20480.58 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 185 |
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| Sequence: | MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
|
|
|
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| BDBM46286 |
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| n/a |
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| Name | BDBM46286 |
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| Synonyms: | (4E)-4-[[[4-fluoranyl-3-(trifluoromethyl)phenyl]methylamino]-sulfanyl-methylidene]-2-methoxy-cyclohexa-2,5-dien-1-one | (4E)-4-[[[4-fluoro-3-(trifluoromethyl)benzyl]amino]-mercapto-methylene]-2-methoxy-cyclohexa-2,5-dien-1-one | (4E)-4-[[[4-fluoro-3-(trifluoromethyl)phenyl]methylamino]-mercaptomethylidene]-2-methoxy-1-cyclohexa-2,5-dienone | (4E)-4-[[[4-fluoro-3-(trifluoromethyl)phenyl]methylamino]-sulfanylmethylidene]-2-methoxycyclohexa-2,5-dien-1-one | MLS-0425623.0001 | cid_44229072 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H13F4NO2S |
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| Mol. Mass. | 359.339 |
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| SMILES | COc1cc(ccc1O)C(=S)NCc1ccc(F)c(c1)C(F)(F)F |
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| Structure | 
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