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TargetDual specificity protein phosphatase 3
LigandBDBM46233
Substrate/Competitorn/a
Meas. Tech.SAR VHR1 absorbance Assay for In Vitro dose response studies.
IC50>100000±n/a nM
Citation PubChem, PC SAR VHR1 absorbance Assay for In Vitro dose response studies. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Dual specificity protein phosphatase 3
Name:Dual specificity protein phosphatase 3
Synonyms:DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR
Type:Hydrolase
Mol. Mass.:20480.58
Organism:Homo sapiens (Human)
Description:n/a
Residue:185
Sequence:
MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
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BDBM46233
n/a
NameBDBM46233
Synonyms:(4E)-4-[(4-ethyl-1-piperazinyl)-mercaptomethylidene]-2-methoxy-1-cyclohexa-2,5-dienone | (4E)-4-[(4-ethylpiperazin-1-yl)-sulfanyl-methylidene]-2-methoxy-cyclohexa-2,5-dien-1-one | (4E)-4-[(4-ethylpiperazin-1-yl)-sulfanylmethylidene]-2-methoxycyclohexa-2,5-dien-1-one | (4E)-4-[(4-ethylpiperazino)-mercapto-methylene]-2-methoxy-cyclohexa-2,5-dien-1-one | MLS-0412088.0001 | cid_5922812
TypeSmall organic molecule
Emp. Form.C14H20N2O2S
Mol. Mass.280.386
SMILESCCN1CCN(CC1)C(=S)c1ccc(O)c(OC)c1
Structure
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