| Reaction Details |
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 | Report a problem with these data |
| Target | D(1B) dopamine receptor |
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| Ligand | BDBM40336 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen |
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| EC50 | 0.00125±n/a nM |
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| Citation |  PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| D(1B) dopamine receptor |
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| Name: | D(1B) dopamine receptor |
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| Synonyms: | D(5) dopamine receptor | D1beta dopamine receptor | DOPAMINE D5 | DRD1B | DRD1L2 | DRD5 | DRD5_HUMAN | dopamine receptor D5 |
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| Type: | Protein |
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| Mol. Mass.: | 52943.41 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21918 |
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| Residue: | 477 |
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| Sequence: | MLPPGSNGTAYPGQFALYQQLAQGNAVGGSAGAPPLGPSQVVTACLLTLLIIWTLLGNVL
VCAAIVRSRHLRANMTNVFIVSLAVSDLFVALLVMPWKAVAEVAGYWPFGAFCDVWVAFD
IMCSTASILNLCVISVDRYWAISRPFRYKRKMTQRMALVMVGLAWTLSILISFIPVQLNW
HRDQAASWGGLDLPNNLANWTPWEEDFWEPDVNAENCDSSLNRTYAISSSLISFYIPVAI
MIVTYTRIYRIAQVQIRRISSLERAAEHAQSCRSSAACAPDTSLRASIKKETKVLKTLSV
IMGVFVCCWLPFFILNCMVPFCSGHPEGPPAGFPCVSETTFDVFVWFGWANSSLNPVIYA
FNADFQKVFAQLLGCSHFCSRTPVETVNISNELISYNQDIVFHKEIAAAYIHMMPNAVTP
GNREVDNDEEEGPFDRMFQIYQTSPDGDPVAESVWELDCEGEISLDKITPFTPNGFH
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| BDBM40336 |
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| n/a |
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| Name | BDBM40336 |
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| Synonyms: | 6-Amino-4-isopropyl-3-thiophen-2-yl-2,4-dihydro-pyrano[2,3-c]pyrazole-5-carbonitrile | 6-amino-4-isopropyl-3-(2-thienyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile | 6-amino-4-propan-2-yl-3-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile | 6-azanyl-4-propan-2-yl-3-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile | MLS000033498 | SMR000014022 | cid_652353 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H14N4OS |
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| Mol. Mass. | 286.352 |
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| SMILES | CC(C)C1C(C#N)C(=N)Oc2[nH]nc(-c3cccs3)c12 |
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| Structure | 
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