| Reaction Details |
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 | Report a problem with these data |
| Target | D(1B) dopamine receptor |
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| Ligand | BDBM48940 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen |
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| EC50 | 0.00817±n/a nM |
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| Citation |  PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| D(1B) dopamine receptor |
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| Name: | D(1B) dopamine receptor |
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| Synonyms: | D(5) dopamine receptor | D1beta dopamine receptor | DOPAMINE D5 | DRD1B | DRD1L2 | DRD5 | DRD5_HUMAN | dopamine receptor D5 |
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| Type: | Protein |
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| Mol. Mass.: | 52943.41 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21918 |
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| Residue: | 477 |
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| Sequence: | MLPPGSNGTAYPGQFALYQQLAQGNAVGGSAGAPPLGPSQVVTACLLTLLIIWTLLGNVL
VCAAIVRSRHLRANMTNVFIVSLAVSDLFVALLVMPWKAVAEVAGYWPFGAFCDVWVAFD
IMCSTASILNLCVISVDRYWAISRPFRYKRKMTQRMALVMVGLAWTLSILISFIPVQLNW
HRDQAASWGGLDLPNNLANWTPWEEDFWEPDVNAENCDSSLNRTYAISSSLISFYIPVAI
MIVTYTRIYRIAQVQIRRISSLERAAEHAQSCRSSAACAPDTSLRASIKKETKVLKTLSV
IMGVFVCCWLPFFILNCMVPFCSGHPEGPPAGFPCVSETTFDVFVWFGWANSSLNPVIYA
FNADFQKVFAQLLGCSHFCSRTPVETVNISNELISYNQDIVFHKEIAAAYIHMMPNAVTP
GNREVDNDEEEGPFDRMFQIYQTSPDGDPVAESVWELDCEGEISLDKITPFTPNGFH
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| BDBM48940 |
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| n/a |
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| Name | BDBM48940 |
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| Synonyms: | (4-oxidanylidene-1,2,3-benzotriazin-3-yl)methyl 1-thiophen-2-ylsulfonylpiperidine-4-carboxylate | (4-oxo-1,2,3-benzotriazin-3-yl)methyl 1-thiophen-2-ylsulfonylpiperidine-4-carboxylate | 1-(2-thienylsulfonyl)isonipecotic acid (4-keto-1,2,3-benzotriazin-3-yl)methyl ester | 1-thiophen-2-ylsulfonyl-4-piperidinecarboxylic acid (4-oxo-1,2,3-benzotriazin-3-yl)methyl ester | MLS000053510 | SMR000063603 | cid_2121421 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H18N4O5S2 |
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| Mol. Mass. | 434.489 |
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| SMILES | O=C(OCn1nnc2ccccc2c1=O)C1CCN(CC1)S(=O)(=O)c1cccs1 |
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| Structure | 
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