| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM48999 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Allosteric Modulators of D1 Receptors: Dose-dependent Assay |
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| EC50 | 0.00365±n/a nM |
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| Citation |  PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Assay PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | DA D1 receptor | DOPAMINE D1 | DRD1 | DRD1_HUMAN | Dopamine D1 receptor | Dopamine D1 receptor (D1R) | Dopamine D1A |
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| Type: | Enzyme |
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| Mol. Mass.: | 49303.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21728 |
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| Residue: | 446 |
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| Sequence: | MRTLNTSAMDGTGLVVERDFSVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTN
FFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVD
RYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNATSLA
ETIDNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKN
CQTTTGNGKPVECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCGS
GETQPFCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPATNNAIET
VSINNNGAAMFSSHHEPRGSISKECNLVYLIPHAVGSSEDLKKEEAAGIARPLEKLSPAL
SVILDYDTDVSLEKIQPITQNGQHPT
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| BDBM48999 |
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| n/a |
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| Name | BDBM48999 |
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| Synonyms: | 2-[3-(2-Chloro-benzyl)-5-cyclopropyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-ylamino]-ethanol | 2-[[3-(2-chlorobenzyl)-5-cyclopropyl-triazolo[4,5-d]pyrimidin-7-yl]amino]ethanol | 2-[[3-[(2-chlorophenyl)methyl]-5-cyclopropyl-7-triazolo[4,5-d]pyrimidinyl]amino]ethanol | 2-[[3-[(2-chlorophenyl)methyl]-5-cyclopropyl-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]amino]ethanol | 2-[[3-[(2-chlorophenyl)methyl]-5-cyclopropyltriazolo[4,5-d]pyrimidin-7-yl]amino]ethanol | MLS000075673 | SMR000007891 | cid_655125 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H17ClN6O |
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| Mol. Mass. | 344.799 |
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| SMILES | OCCNc1nc(nc2n(Cc3ccccc3Cl)nnc12)C1CC1 |
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| Structure | 
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