Reaction Details |
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Target | Ras-related C3 botulinum toxin substrate 1 |
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Ligand | BDBM54675 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype |
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Ki | 250±n/a nM |
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Citation | PubChem, PC Additional SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 wildtype PubChem Bioassay(2009)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Ras-related C3 botulinum toxin substrate 1 |
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Name: | Ras-related C3 botulinum toxin substrate 1 |
Synonyms: | RAC1_MOUSE | Rac1 | Rac1 protein |
Type: | PROTEIN |
Mol. Mass.: | 21455.91 |
Organism: | Mus musculus |
Description: | EBI_101485 |
Residue: | 192 |
Sequence: | MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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BDBM54675 |
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n/a |
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Name | BDBM54675 |
Synonyms: | (5Z)-5-(2-ketoindolin-3-ylidene)hydantoin | (5Z)-5-(2-oxidanylidene-1H-indol-3-ylidene)imidazolidine-2,4-dione | (5Z)-5-(2-oxo-1H-indol-3-ylidene)imidazolidine-2,4-dione | UNM-0000305761 | cid_15716919 |
Type | Small organic molecule |
Emp. Form. | C11H7N3O3 |
Mol. Mass. | 229.1916 |
SMILES | O=C1NC(=O)\C(N1)=C1\C(=O)Nc2ccccc12 |
Structure |
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