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TargetStreptokinase A
LigandBDBM58086
Substrate/Competitorn/a
Meas. Tech.Absorbance Microorganism-Based Dose Response HTS to Identify Inhibitors of Streptokinase Expression
EC50 150000±n/a nM
Citation PubChem, PC Absorbance Microorganism-Based Dose Response HTS to Identify Inhibitors of Streptokinase Expression PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Streptokinase A
Name:Streptokinase A
Synonyms:STRP_STRP1 | ska | streptokinase A precursor
Type:Enzyme Catalytic Domain
Mol. Mass.:49924.80
Organism:Streptococcus pyogenes M1 GAS
Description:gi_15675770
Residue:440
Sequence:
MKNYLSIGVIALLFALTFGTVKSVQAIAGYGWLPDRPPINNSQLVVSMAGIVEGTDKKVF
INFFEIDLTSQPAHGGKTEQGLSPKSKPFATDNGAMPHKLEKADLLKAIQKQLIANVHSN
DGYFEVIDFASDATITDRNGKVYFADKDGSVTLPTQPVQEFLLKGHVRVRPYKEKPVQNQ
AKSVDVEYTVQFTPLNPDDDFRPGLKDTKLLKTLAIGDTITSQELLAQAQSILNKTHPGY
TIYERDSSIVTHDNDIFRTILPMDQEFTYHVKNREQAYEINPKTGIKEKTNNTDLVSEKY
YVLKQGEKPYDPFDRSHLKLFTIKYVDVNTNELLKSEQLLTASERNLDFRDLYDPRDKAK
LLYNNLDAFDIMDYTLTGKVEDNHDKNNRVVTVYMGKRPKGAKGSYHLAYDKDLYTEEER
KAYSYLRDTGTPIPDNPKDK
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  Blast E-value cutoff:
BDBM58086
n/a
NameBDBM58086
Synonyms:MLS000806923 | SMR000414723 | Tricyclo[4.3.1.1*3,8*]undecane-1-carboxylic acid [1-(3-bromo-2-hydroxy-5-nitro-phenyl)-meth-(E)-ylidene]-hydrazide | cid_6291459
TypeSmall organic molecule
Emp. Form.C19H22BrN3O4
Mol. Mass.436.3
SMILES[H]C12CC3([H])CC(C1)(CC([H])(C2)CC3)C(=O)NN\C=C1/C=C(C=C(Br)C1=O)[N+]([O-])=O |c:23,t:25,TLB:12:9:7:3.5.2,THB:2:1:8:3.5.12.13,2:3:8:1.7.11,13:3:7:9.8.11|
Structure
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