| Reaction Details |
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 | Report a problem with these data |
| Target | M17 leucyl aminopeptidase |
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| Ligand | BDBM60125 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) |
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| IC50 | 1000±n/a nM |
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| Citation |  PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| M17 leucyl aminopeptidase |
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| Name: | M17 leucyl aminopeptidase |
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| Synonyms: | leucine aminopeptidase |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 67834.32 |
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| Organism: | Plasmodium falciparum 3D7 |
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| Description: | gi_124809582 |
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| Residue: | 605 |
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| Sequence: | MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
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| BDBM60125 |
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| n/a |
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| Name | BDBM60125 |
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| Synonyms: | 1,2,3,4,7,7-hexachloro-6-(p-phenetylcarbamoyl)bicyclo[2.2.1]hept-2-ene-5-carboxylic acid | 1,2,3,4,7,7-hexachloro-6-[(4-ethoxyanilino)-oxomethyl]-5-bicyclo[2.2.1]hept-2-enecarboxylic acid | 1,2,3,4,7,7-hexachloro-6-[(4-ethoxyphenyl)carbamoyl]bicyclo[2.2.1]hept-2-ene-5-carboxylic acid | 1,2,3,4,7,7-hexakis(chloranyl)-6-[(4-ethoxyphenyl)carbamoyl]bicyclo[2.2.1]hept-2-ene-5-carboxylic acid | MLS000713583 | SMR000273064 | cid_3122377 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H13Cl6NO4 |
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| Mol. Mass. | 508.007 |
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| SMILES | CCOc1ccc(NC(=O)C2C(C(O)=O)C3(Cl)C(Cl)=C(Cl)C2(Cl)C3(Cl)Cl)cc1 |t:18,TLB:8:10:23:19.17,20:19:10.11:23,THB:12:11:23:19.17,18:17:10.11:23| |
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| Structure | 
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