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TargetNeuropeptide Y receptor type 1
LigandBDBM61791
Substrate/Competitorn/a
Meas. Tech.Fluorescence-based dose response cell-based high-throughput screening assay for agonists of NPY-Y1.
EC50 11619±n/a nM
Citation PubChem, PC Fluorescence-based dose response cell-based high-throughput screening assay for agonists of NPY-Y1. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Neuropeptide Y receptor type 1
Name:Neuropeptide Y receptor type 1
Synonyms:NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1
Type:Enzyme Catalytic Domain
Mol. Mass.:44399.07
Organism:Homo sapiens (Human)
Description:NPY-Y1 NPY1R HUMAN::P25929
Residue:384
Sequence:
MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLA
LIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQ
CVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMT
DEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKR
RNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNL
LFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVS
KTSLKQASPVAFKKINNNDDNEKI
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  Blast E-value cutoff:
BDBM61791
n/a
NameBDBM61791
Synonyms:1-(4-chloranylphenoxy)-3-(2,3-dihydro-1H-inden-2-ylamino)propan-2-ol | 1-(4-chlorophenoxy)-3-(2,3-dihydro-1H-inden-2-ylamino)-2-propanol | 1-(4-chlorophenoxy)-3-(2,3-dihydro-1H-inden-2-ylamino)propan-2-ol | 1-(4-chlorophenoxy)-3-(indan-2-ylamino)propan-2-ol | MLS000830157 | SMR000458078 | cid_2809885
TypeSmall organic molecule
Emp. Form.C18H20ClNO2
Mol. Mass.317.81
SMILESOC(CNC1Cc2ccccc2C1)COc1ccc(Cl)cc1
Structure
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