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TargetNeuropeptide Y receptor type 2
LigandBDBM61778
Substrate/Competitorn/a
Meas. Tech.Fluorescence-based counterscreen for agonists of NPY-Y1: cell-based high-throughput dose response assay for agonists of NPY-Y2.
EC50 12439±n/a nM
Citation PubChem, PC Fluorescence-based counterscreen for agonists of NPY-Y1: cell-based high-throughput dose response assay for agonists of NPY-Y2. PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Neuropeptide Y receptor type 2
Name:Neuropeptide Y receptor type 2
Synonyms:NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:Enzyme Catalytic Domain
Mol. Mass.:42734.65
Organism:Homo sapiens (Human)
Description:NPY-Y2 NPY2R HUMAN::P49146
Residue:381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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BDBM61778
n/a
NameBDBM61778
Synonyms:2-benzyl-3-[4-(diethylamino)anilino]-3-keto-propionic acid ethyl ester | 3-[4-(diethylamino)anilino]-3-oxo-2-(phenylmethyl)propanoic acid ethyl ester | MLS000573081 | SMR000185011 | cid_2836861 | ethyl 2-benzyl-3-[4-(diethylamino)anilino]-3-oxopropanoate | ethyl 2-benzyl-3-{[4-(diethylamino)phenyl]amino}-3-oxopropanoate | ethyl 3-[[4-(diethylamino)phenyl]amino]-3-oxidanylidene-2-(phenylmethyl)propanoate
TypeSmall organic molecule
Emp. Form.C22H28N2O3
Mol. Mass.368.4693
SMILESCCOC(=O)C(Cc1ccccc1)C(=O)Nc1ccc(cc1)N(CC)CC
Structure
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