| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 2 |
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| Ligand | BDBM34803 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence-based counterscreen for agonists of NPY-Y1: cell-based high-throughput dose response assay for agonists of NPY-Y2. |
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| EC50 | 19286±n/a nM |
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| Citation |  PubChem, PC Fluorescence-based counterscreen for agonists of NPY-Y1: cell-based high-throughput dose response assay for agonists of NPY-Y2. PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Neuropeptide Y receptor type 2 |
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| Name: | Neuropeptide Y receptor type 2 |
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| Synonyms: | NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 42734.65 |
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| Organism: | Homo sapiens (Human) |
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| Description: | NPY-Y2 NPY2R HUMAN::P49146 |
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| Residue: | 381 |
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| Sequence: | MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
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| BDBM34803 |
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| n/a |
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| Name | BDBM34803 |
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| Synonyms: | (4E)-2,3-dihydroxy-4-[[[2-(2-methoxyethylimino)-4-(2-thienyl)-4-thiazolin-3-yl]amino]methylene]cyclohexa-2,5-dien-1-one | (4E)-2,3-dihydroxy-4-[[[2-(2-methoxyethylimino)-4-thiophen-2-yl-1,3-thiazol-3-yl]amino]methylidene]cyclohexa-2,5-dien-1-one | (4E)-2,3-dihydroxy-4-[[[2-(2-methoxyethylimino)-4-thiophen-2-yl-3-thiazolyl]amino]methylidene]-1-cyclohexa-2,5-dienone | (4E)-4-[[[2-(2-methoxyethylimino)-4-thiophen-2-yl-1,3-thiazol-3-yl]amino]methylidene]-2,3-bis(oxidanyl)cyclohexa-2,5-dien-1-one | MLS000339614 | SMR000242031 | cid_6146295 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H17N3O4S2 |
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| Mol. Mass. | 391.465 |
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| SMILES | COCCN=c1scc(-c2cccs2)n1N=Cc1ccc(O)c(O)c1O |w:15.16,4.3| |
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| Structure | 
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