| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM62197 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay |
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| EC50 | >32000±n/a nM |
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| Citation |  PubChem, PC SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40382.98 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor. |
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| Residue: | 372 |
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| Sequence: | MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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| BDBM62197 |
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| n/a |
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| Name | BDBM62197 |
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| Synonyms: | (phenylmethyl) N-[1-[(3-bromophenyl)carbamothioylamino]-2,2,2-tris(chloranyl)ethyl]carbamate | MLS-0425698.0001 | N-[1-[(3-bromophenyl)thiocarbamoylamino]-2,2,2-trichloro-ethyl]carbamic acid benzyl ester | N-[1-[[(3-bromoanilino)-sulfanylidenemethyl]amino]-2,2,2-trichloroethyl]carbamic acid (phenylmethyl) ester | benzyl N-[1-[(3-bromophenyl)carbamothioylamino]-2,2,2-trichloroethyl]carbamate | cid_3091269 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H15BrCl3N3O2S |
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| Mol. Mass. | 511.648 |
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| SMILES | ClC(Cl)(Cl)C(NC(=O)OCc1ccccc1)NC(=S)Nc1cccc(Br)c1 |
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| Structure | 
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