| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM54785 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay |
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| EC50 | >32000±n/a nM |
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| Citation |  PubChem, PC SAR Analysis of Agonists of the DOR Receptor using an Image-Based Assay PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | D-OR-1 | DOR-1 | Delta opioid receptor | Delta-type opioid receptor (Delta) | OPIATE Delta | OPRD | OPRD1 | OPRD_HUMAN | OPRK1 | opioid receptor, delta 1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40382.98 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Competition binding assays were carried out using membrane preparations from transfected HN9.10 cells that constitutively expressed the delta opioid receptor. |
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| Residue: | 372 |
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| Sequence: | MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTAC
TPSDGPGGGAAA
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|
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| BDBM54785 |
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| n/a |
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| Name | BDBM54785 |
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| Synonyms: | MLS000729763 | N-[1-(cyclopentylamino)-2-methyl-1-oxidanylidene-butan-2-yl]-N-(thiophen-2-ylmethyl)pyridine-2-carboxamide | N-[1-(cyclopentylamino)-2-methyl-1-oxobutan-2-yl]-N-(thiophen-2-ylmethyl)-2-pyridinecarboxamide | N-[1-(cyclopentylamino)-2-methyl-1-oxobutan-2-yl]-N-(thiophen-2-ylmethyl)pyridine-2-carboxamide | N-[1-(cyclopentylcarbamoyl)-1-methyl-propyl]-N-(2-thenyl)picolinamide | SMR000308040 | Structure possibly contains amino acid derivative which is not supported in current version! | cid_3950572 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H27N3O2S |
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| Mol. Mass. | 385.523 |
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| SMILES | CCC(C)(N(Cc1cccs1)C(=O)c1ccccn1)C(=O)NC1CCCC1 |
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| Structure | 
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