Ki Summary

Reaction Details

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Target

Serine/threonine-protein phosphatase PP1-alpha catalytic subunit

Ligand

BDBM64779

Substrate/Competitor

n/a

Meas. Tech.

Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput dose response assay for inhibitors of Protein Phosphatase 1 (PP1)

IC50

67047±n/a nM

Citation

PubChem, PC Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput dose response assay for inhibitors of Protein Phosphatase 1 (PP1) PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Serine/threonine-protein phosphatase PP1-alpha catalytic subunit

Name:

Serine/threonine-protein phosphatase PP1-alpha catalytic subunit

Synonyms:

Type:

PROTEIN

Mol. Mass.:

37510.66

Organism:

Homo sapiens (Human)

Description:

ChEMBL_197827

Residue:

330

Sequence:

MSDSEKLNLDSIIGRLLEVQGSRPGKNVQLTENEIRGLCLKSREIFLSQPILLELEAPLK
ICGDIHGQYYDLLRLFEYGGFPPESNYLFLGDYVDRGKQSLETICLLLAYKIKYPENFFL
LRGNHECASINRIYGFYDECKRRYNIKLWKTFTDCFNCLPIAAIVDEKIFCCHGGLSPDL
QSMEQIRRIMRPTDVPDQGLLCDLLWSDPDKDVQGWGENDRGVSFTFGAEVVAKFLHKHD
LDLICRAHQVVEDGYEFFAKRQLVTLFSAPNYCGEFDNAGAMMSVDETLMCSFQILKPAD
KNKGKYGQFSGLNPGGRPITPPRNSAKAKK

BDBM64779

n/a

Name

BDBM64779

Synonyms:

(6Z)-6-(1,2-dihydro-1,2,3,4-tetrazol-5-ylidene)-4-nitro-cyclohexa-2,4-dien-1-one | (6Z)-6-(1,2-dihydrotetrazol-5-ylidene)-4-nitro-1-cyclohexa-2,4-dienone | (6Z)-6-(1,2-dihydrotetrazol-5-ylidene)-4-nitro-cyclohexa-2,4-dien-1-one | (6Z)-6-(1,2-dihydrotetrazol-5-ylidene)-4-nitrocyclohexa-2,4-dien-1-one | 4-nitro-2-(2H-tetraazol-5-yl)phenol | MLS000540078 | SMR000162423 | cid_11839800

Type

Small organic molecule

Emp. Form.

C7H5N5O3

Mol. Mass.

207.1463

SMILES

[O-][N+](=O)c1ccc(=O)[c-](c1)-c1[nH]nn[nH+]1

Structure