Ki Summary

Reaction Details

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Target

Serine/threonine-protein phosphatase PP1-alpha catalytic subunit

Ligand

BDBM61210

Substrate/Competitor

n/a

Meas. Tech.

Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput dose response assay for inhibitors of Protein Phosphatase 1 (PP1)

IC50

67047±n/a nM

Citation

PubChem, PC Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput dose response assay for inhibitors of Protein Phosphatase 1 (PP1) PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Serine/threonine-protein phosphatase PP1-alpha catalytic subunit

Name:

Serine/threonine-protein phosphatase PP1-alpha catalytic subunit

Synonyms:

Type:

PROTEIN

Mol. Mass.:

37510.66

Organism:

Homo sapiens (Human)

Description:

ChEMBL_197827

Residue:

330

Sequence:

MSDSEKLNLDSIIGRLLEVQGSRPGKNVQLTENEIRGLCLKSREIFLSQPILLELEAPLK
ICGDIHGQYYDLLRLFEYGGFPPESNYLFLGDYVDRGKQSLETICLLLAYKIKYPENFFL
LRGNHECASINRIYGFYDECKRRYNIKLWKTFTDCFNCLPIAAIVDEKIFCCHGGLSPDL
QSMEQIRRIMRPTDVPDQGLLCDLLWSDPDKDVQGWGENDRGVSFTFGAEVVAKFLHKHD
LDLICRAHQVVEDGYEFFAKRQLVTLFSAPNYCGEFDNAGAMMSVDETLMCSFQILKPAD
KNKGKYGQFSGLNPGGRPITPPRNSAKAKK

BDBM61210

n/a

Name

BDBM61210

Synonyms:

3-Acetyl-3a,8b-dihydroxy-2-methyl-3a,8b-dihydro-indeno[1,2-b]furan-4-one | 3-acetyl-3a,8b-dihydroxy-2-methyl-4-indeno[1,2-b]furanone | 3-acetyl-3a,8b-dihydroxy-2-methyl-indeno[1,2-b]furan-4-one | 3-acetyl-3a,8b-dihydroxy-2-methylindeno[1,2-b]furan-4-one | 3-ethanoyl-2-methyl-3a,8b-bis(oxidanyl)indeno[1,2-b]furan-4-one | MLS000768249 | SMR000431570 | cid_2828331

Type

Small organic molecule

Emp. Form.

C14H12O5

Mol. Mass.

260.2421

SMILES

CC(=O)C1=C(C)OC2(O)c3ccccc3C(=O)C12O |c:3|

Structure