| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM62190 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | SAR Analysis of Antagonists of the MOR Receptor using an Image-Based Assay |
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| IC50 | >32000±n/a nM |
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| Citation |  PubChem, PC SAR Analysis of Antagonists of the MOR Receptor using an Image-Based Assay PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 44789.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35372 |
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| Residue: | 400 |
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| Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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|
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| BDBM62190 |
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| n/a |
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| Name | BDBM62190 |
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| Synonyms: | 4-[[(4-acetylphenyl)sulfonylamino]methyl]-N-[2-(3-fluoroanilino)-2-keto-ethyl]-N-methyl-benzamide | 4-[[(4-acetylphenyl)sulfonylamino]methyl]-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methylbenzamide | 4-[[(4-ethanoylphenyl)sulfonylamino]methyl]-N-[2-[(3-fluorophenyl)amino]-2-oxidanylidene-ethyl]-N-methyl-benzamide | MLS-0332830.0001 | cid_16295215 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H24FN3O5S |
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| Mol. Mass. | 497.539 |
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| SMILES | CN(CC(=O)Nc1cccc(F)c1)C(=O)c1ccc(CNS(=O)(=O)c2ccc(cc2)C(C)=O)cc1 |
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| Structure | 
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