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TargetTrans-activator protein BZLF1
LigandBDBM64862
Substrate/Competitorn/a
Meas. Tech.Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50 47562±n/a nM
Citation PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Trans-activator protein BZLF1
Name:Trans-activator protein BZLF1
Synonyms:BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:Enzyme Catalytic Domain
Mol. Mass.:26856.37
Organism:Human herpesvirus 4
Description:gi_82503229
Residue:245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQ
LTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNS
TVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRY
KNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHE
DLLNF
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  Blast E-value cutoff:
BDBM64862
n/a
NameBDBM64862
Synonyms:5-chloranyl-7-[(4-methylpiperazin-1-yl)-pyridin-2-yl-methyl]quinolin-8-ol | 5-chloro-7-[(4-methyl-1-piperazinyl)-(2-pyridinyl)methyl]-8-quinolinol | 5-chloro-7-[(4-methylpiperazin-1-yl)-pyridin-2-ylmethyl]quinolin-8-ol | 5-chloro-7-[(4-methylpiperazino)-(2-pyridyl)methyl]quinolin-8-ol | MLS000774453 | SMR000371742 | cid_3515733
TypeSmall organic molecule
Emp. Form.C20H21ClN4O
Mol. Mass.368.86
SMILESCN1CCN(CC1)C(c1ccccn1)c1cc(Cl)c2cccnc2c1O
Structure
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