Ki Summary

Reaction Details

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Target

Heat shock factor protein 1

Ligand

BDBM72271

Substrate/Competitor

n/a

Meas. Tech.

Luminescence Cell-Based Dose Retest to Identify Potentiators of Heat Shock Factor 1 (HSF1)

EC50

>260000±n/a nM

Citation

PubChem, PC Luminescence Cell-Based Dose Retest to Identify Potentiators of Heat Shock Factor 1 (HSF1) PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Heat shock factor protein 1

Name:

Heat shock factor protein 1

Synonyms:

HSF1_MOUSE | Hsf1 | Hsf1 protein

Type:

Enzyme Catalytic Domain

Mol. Mass.:

57208.68

Organism:

Mus musculus

Description:

P38532

Residue:

525

Sequence:

MDLAVGPGAAGPSNVPAFLTKLWTLVSDPDTDALICWSPSGNSFHVFDQGQFAKEVLPKY
FKHNNMASFVRQLNMYGFRKVVHIEQGGLVKPERDDTEFQHPCFLRGQEQLLENIKRKVT
SVSTLKSEDIKIRQDSVTRLLTDVQLMKGKQECMDSKLLAMKHENEALWREVASLRQKHA
QQQKVVNKLIQFLISLVQSNRILGVKRKIPLMLSDSNSAHSVPKYGRQYSLEHVHGPGPY
SAPSPAYSSSSLYSSDAVTSSGPIISDITELAPTSPLASPGRSIDERPLSSSTLVRVKQE
PPSPPHSPRVLEASPGRPSSMDTPLSPTAFIDSILRESEPTPAASNTAPMDTTGAQAPAL
PTPSTPEKCLSVACLDKNELSDHLDAMDSNLDNLQTMLTSHGFSVDTSALLDLFSPSVTM
PDMSLPDLDSSLASIQELLSPQEPPRPIEAENSNPDSGKQLVHYTAQPLFLLDPDAVDTG
SSELPVLFELGESSYFSEGDDYTDDPTISLLTGTEPHKAKDPTVS

BDBM72271

n/a

Name

BDBM72271

Synonyms:

2-(1-naphthalenylamino)-N-[(4-nitrophenyl)methylideneamino]acetamide | 2-(1-naphthylamino)-N'-[(1E)-(4-nitrophenyl)methylene]acetohydrazide | 2-(1-naphthylamino)-N-[(4-nitrobenzylidene)amino]acetamide | 2-(1-naphthylamino)-N-[(E)-(4-nitrobenzylidene)amino]acetamide | 2-(naphthalen-1-ylamino)-N-[(4-nitrophenyl)methylideneamino]acetamide | 2-(naphthalen-1-ylamino)-N-[(4-nitrophenyl)methylideneamino]ethanamide | MLS000584418 | SMR000203581 | cid_684162

Type

Small organic molecule

Emp. Form.

C19H16N4O3

Mol. Mass.

348.3553

SMILES

[O-][N+](=O)c1ccc(\C=N\NC(=O)CNc2cccc3ccccc23)cc1

Structure