| Reaction Details |
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 | Report a problem with these data |
| Target | Heat shock factor protein 1 |
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| Ligand | BDBM72275 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Luminescence Cell-Based Dose Retest to Identify Potentiators of Heat Shock Factor 1 (HSF1) |
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| EC50 | 13400±n/a nM |
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| Citation |  PubChem, PC Luminescence Cell-Based Dose Retest to Identify Potentiators of Heat Shock Factor 1 (HSF1) PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Heat shock factor protein 1 |
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| Name: | Heat shock factor protein 1 |
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| Synonyms: | HSF1_MOUSE | Hsf1 | Hsf1 protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 57208.68 |
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| Organism: | Mus musculus |
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| Description: | P38532 |
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| Residue: | 525 |
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| Sequence: | MDLAVGPGAAGPSNVPAFLTKLWTLVSDPDTDALICWSPSGNSFHVFDQGQFAKEVLPKY
FKHNNMASFVRQLNMYGFRKVVHIEQGGLVKPERDDTEFQHPCFLRGQEQLLENIKRKVT
SVSTLKSEDIKIRQDSVTRLLTDVQLMKGKQECMDSKLLAMKHENEALWREVASLRQKHA
QQQKVVNKLIQFLISLVQSNRILGVKRKIPLMLSDSNSAHSVPKYGRQYSLEHVHGPGPY
SAPSPAYSSSSLYSSDAVTSSGPIISDITELAPTSPLASPGRSIDERPLSSSTLVRVKQE
PPSPPHSPRVLEASPGRPSSMDTPLSPTAFIDSILRESEPTPAASNTAPMDTTGAQAPAL
PTPSTPEKCLSVACLDKNELSDHLDAMDSNLDNLQTMLTSHGFSVDTSALLDLFSPSVTM
PDMSLPDLDSSLASIQELLSPQEPPRPIEAENSNPDSGKQLVHYTAQPLFLLDPDAVDTG
SSELPVLFELGESSYFSEGDDYTDDPTISLLTGTEPHKAKDPTVS
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| BDBM72275 |
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| n/a |
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| Name | BDBM72275 |
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| Synonyms: | (E)-2-butenedioic acid O4-[2-[(diphenylmethyl)amino]-2-oxoethyl] ester O1-ethyl ester | (E)-but-2-enedioic acid O4-[2-(benzhydrylamino)-2-keto-ethyl] ester O1-ethyl ester | 4-O-[2-(benzhydrylamino)-2-oxoethyl] 1-O-ethyl (E)-but-2-enedioate | MLS000374880 | O4-[2-[(diphenylmethyl)amino]-2-oxidanylidene-ethyl] O1-ethyl (E)-but-2-enedioate | SMR000254234 | cid_5889878 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H21NO5 |
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| Mol. Mass. | 367.3951 |
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| SMILES | CCOC(=O)\C=C\C(=O)OCC(=O)NC(c1ccccc1)c1ccccc1 |
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| Structure | 
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