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TargetNeuropeptides B/W receptor type 1
LigandBDBM75883
Substrate/Competitorn/a
Meas. Tech.Late-stage fluorescence-based dose response cell-based screening assay to identify antagonists of the G-protein coupled receptor 7 (GPR7)
IC50 2200±n/a nM
Citation PubChem, PC Late-stage fluorescence-based dose response cell-based screening assay to identify antagonists of the G-protein coupled receptor 7 (GPR7) PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Neuropeptides B/W receptor type 1
Name:Neuropeptides B/W receptor type 1
Synonyms:GPR7 | NPBW1_HUMAN | NPBWR1 | neuropeptides B/W receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:36111.82
Organism:Homo sapiens (Human)
Description:gi_119607128
Residue:328
Sequence:
MDNASFSEPWPANASGPDPALSCSNASTLAPLPAPLAVAVPVVYAVICAVGLAGNSAVLY
VLLRAPRMKTVTNLFILNLAIADELFTLVLPINIADFLLRQWPFGELMCKLIVAIDQYNT
FSSLYFLTVMSADRYLVVLATAESRRVAGRTYSAARAVSLAVWGIVTLVVLPFAVFARLD
DEQGRRQCVLVFPQPEAFWWRASRLYTLVLGFAIPVSTICVLYTTLLCRLHAMRLDSHAK
ALERAKKRVTFLVVAILAVCLLCWTPYHLSTVVALTTDLPQTPLVIAISYFITSLSYANS
CLNPFLYAFLDASFRRNLRQLITCRAAA
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  Blast E-value cutoff:
BDBM75883
n/a
NameBDBM75883
Synonyms:5-chloranyl-2-(4-methylphenyl)-4-[4-(trifluoromethyl)phenoxy]pyridazin-3-one | 5-chloro-2-(4-methylphenyl)-4-[4-(trifluoromethyl)phenoxy]-3-pyridazinone | 5-chloro-2-(4-methylphenyl)-4-[4-(trifluoromethyl)phenoxy]pyridazin-3-one | 5-chloro-2-(p-tolyl)-4-[4-(trifluoromethyl)phenoxy]pyridazin-3-one | SR-02000000351 | SR-02000000351-1 | cid_46172942
TypeSmall organic molecule
Emp. Form.C18H12ClF3N2O2
Mol. Mass.380.748
SMILESCc1ccc(cc1)-n1ncc(Cl)c(Oc2ccc(cc2)C(F)(F)F)c1=O
Structure
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